Research map: Design of sunflower trypsin inhibitor 1 derived probes targeting the LDLR and evaluation of their brain delivery

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  1. The blood-brain barrier: Bottleneck in brain drug development · William M. Pardridge · 2004 · 2810 citations · Cited by this paper
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  25. ANG1005, a Brain-Penetrating Peptide–Drug Conjugate, Shows Activity in Patients with Breast Cancer with Leptomeningeal Carcinomatosis and Recurrent Brain Metastases · Priya Kumthekar · 2020 · 259 citations · Cited by this paper
  26. Designing macrocyclic disulfide-rich peptides for biotechnological applications · Conan K. L. Wang · 2018 · 236 citations · Cited by this paper
  27. A Historical Review of Brain Drug Delivery · William M. Pardridge · 2022 · 228 citations · Cited by this paper
  28. Differential expression of receptors mediating receptor-mediated transcytosis (RMT) in brain microvessels, brain parenchyma and peripheral tissues of the mouse and the human · Wandong Zhang · 2020 · 201 citations · Cited by this paper
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  36. Low-density lipoprotein receptor structure and folding · Jürgen Gent · 2004 · 122 citations · Cited by this paper
  37. Use of LDL receptor—targeting peptide vectors for in vitro and in vivo cargo transport across the blood‐brain barrier · Yves Molino · 2017 · 119 citations · Cited by this paper
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